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| Drug Name | XMU-MP-2 |
| Trade Name | |
| Synonyms | |
| Drug Descriptions |
XMU-MP-2 is a small molecule that inhibits PTK6 (BRK), resulting in decreased downstream signaling and reduced proliferation of PTK6 (BRK)-expressing tumor cells (PMID: 27758886). |
| DrugClasses | |
| CAS Registry Number | 2031152-10-8 |
| NCIT ID | NA |
| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| Afimoxifene + XMU-MP-2 | Afimoxifene XMU-MP-2 | 0 | 0 |
| CP-724,714 + XMU-MP-2 | CP-724,714 XMU-MP-2 | 0 | 0 |
| XMU-MP-2 | XMU-MP-2 | 0 | 0 |