Missing content? – Request curation!
Request curation for specific Genes, Variants, or PubMed publications.
Have questions, comments, or suggestions? - Let us know!
Email us at : ckbsupport@genomenon.com
| Drug Name | GDC-0152 |
| Trade Name | |
| Synonyms | |
| Drug Descriptions |
GDC-0152 is a SMAC mimetic compound, which antagonizes inhibitor of apoptosis proteins (IAPs), resulting in increased apoptosis and differentiation of tumor cells (PMID: 27490930, PMID: 31521127). |
| DrugClasses | SMAC Mimetic 8 |
| CAS Registry Number | 873652-48-3 |
| NCIT ID | C88274 |
| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| GDC-0152 | GDC-0152 | 1 | 0 |