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| Drug Name | EPI-506 |
| Trade Name | |
| Synonyms | Ralaniten acetate |
| Drug Descriptions |
EPI-506 (ralaniten acetate), the prodrug for EPI-002, is a small molecule that inhibits the N-terminal domain of the androgen receptor (AR), potentially resulting in decreased AR signaling, including in the context of mutant AR (PMID: 27628492, PMID: 27140928). |
| DrugClasses | Hormone - Anti-androgens 56 |
| CAS Registry Number | 1637573-04-6 |
| NCIT ID | C124654 |
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| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| EPI-506 | EPI-506 | 0 | 1 |
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