TRC253
Drug Detail
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| Drug Name | TRC253 |
| Trade Name | |
| Synonyms | JNJ-63576253|TRC-253|TRC 253 |
| Drug Descriptions |
TRC253 binds androgen receptor (AR), including wild-type AR and some mutant versions, resulting in decreased receptor activation and downstream signaling, and potentially leading to decreased growth of AR-expressing tumor cells (PMID: 30462924). |
| DrugClasses | Hormone - Anti-androgens 57 |
| CAS Registry Number | 2110426-27-0 |
| NCIT ID | C131874 |
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| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| TRC253 | TRC253 | 0 | 1 |
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