CFI-402257
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| Drug Name | CFI-402257 |
| Trade Name | |
| Synonyms | |
| Drug Descriptions |
CFI-402257 selectively inhibits TTK (MPS1), resulting in chromosomal segregation errors, and potentially leading to decreased tumor cell growth (PMID: 28270606, PMID: 29378962). |
| DrugClasses | MPS1 Inhibitor 27 |
| CAS Registry Number | 1610759-22-2 |
| NCIT ID | C128288 |
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| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| CFI-402257 | CFI-402257 | 0 | 2 |
| CFI-402257 + Fulvestrant | CFI-402257 Fulvestrant | 0 | 1 |
| CFI-402257 + Paclitaxel | CFI-402257 Paclitaxel | 0 | 1 |
| CFI-402257 + unspecified PD-1 antibody | CFI-402257 unspecified PD-1 antibody | 0 | 0 |
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