Selitrectinib
Drug Detail
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| Drug Name | Selitrectinib |
| Trade Name | |
| Synonyms | LOXO-195|BAY 2731954 |
| Drug Descriptions |
Selitrectinib (LOXO-195) is an inhibitor of NTRK1, NTRK2, and NTRK3, which may result in inhibition of tumor growth and tumor regression (PMID: 28578312). |
| DrugClasses | Trk Receptor Inhibitor (Pan) 33 |
| CAS Registry Number | 2097002-61-2 |
| NCIT ID | C138160 |
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| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| Crizotinib + Selitrectinib | Crizotinib Selitrectinib | 0 | 0 |
| Dabrafenib + Selitrectinib + Trametinib | Dabrafenib Selitrectinib Trametinib | 0 | 0 |
| Selitrectinib | Selitrectinib | 0 | 1 |
| Selitrectinib + Trametinib | Selitrectinib Trametinib | 0 | 0 |
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