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Drug Name | TP-0184 |
Trade Name | |
Synonyms | TP0184|TP 0184|itacnosertib |
Drug Descriptions |
TP-0184 inhibits ACVR1 and FLT3 and reduces downstream signaling, potentially resulting in decreased tumor cell proliferation and inhibition of tumor growth (PMID: 38007585). |
DrugClasses | FLT3 Inhibitor 69 |
CAS Registry Number | 1628870-27-8 |
NCIT ID | C156729 |
Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
---|---|---|---|
TP-0184 | TP-0184 | 1 | 2 |
TP-0184 + Venetoclax | TP-0184 Venetoclax | 1 | 0 |