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Gene | IDH1 |
Variant | R132L |
Impact List | missense |
Protein Effect | gain of function |
Gene Variant Descriptions | IDH1 R132L lies within the active site of the Idh1 protein (PMID: 19228619). R132L confers a gain of function to Idh1, as indicated by increased conversion of alpha-ketoglutarate to the onco-metabolite 2HG (R(-)-2-hydroxyglutarate) in cell culture (PMID: 19935646, PMID: 21326614). |
Associated Drug Resistance | |
Category Variants Paths |
IDH1 mutant IDH1 act mut IDH1 R132L IDH1 mutant IDH1 R132X IDH1 R132L |
Transcript | NM_005896.4 |
gDNA | chr2:g.208248388C>A |
cDNA | c.395G>T |
Protein | p.R132L |
Source Database | RefSeq |
Genome Build | GRCh38/hg38 |
Transcript | gDNA | cDNA | Protein | Source Database | Genome Build |
---|---|---|---|---|---|
NM_005896 | chr2:g.208248388C>A | c.395G>T | p.R132L | RefSeq | GRCh38/hg38 |
NM_001282387 | chr2:g.208248388C>A | c.395G>T | p.R132L | RefSeq | GRCh38/hg38 |
NM_005896.3 | chr2:g.208248388C>A | c.395G>T | p.R132L | RefSeq | GRCh38/hg38 |
NM_001282386.1 | chr2:g.208248388C>A | c.395G>T | p.R132L | RefSeq | GRCh38/hg38 |
NM_005896.4 | chr2:g.208248388C>A | c.395G>T | p.R132L | RefSeq | GRCh38/hg38 |
NM_001282386.1 | chr2:g.208248388C>A | c.395G>T | p.R132L | RefSeq | GRCh38/hg38 |
NM_001282387.1 | chr2:g.208248388C>A | c.395G>T | p.R132L | RefSeq | GRCh38/hg38 |
NM_001282386 | chr2:g.208248388C>A | c.395G>T | p.R132L | RefSeq | GRCh38/hg38 |
NM_001282387.1 | chr2:g.208248388C>A | c.395G>T | p.R132L | RefSeq | GRCh38/hg38 |
Clinical Trial | Phase | Therapies | Title | Recruitment Status | Covered Countries | Other Countries |
---|---|---|---|---|---|---|
NCT05876754 | Phase III | Ivosidenib | An Early Access Study of Ivosidenib in Patients With a Pretreated Locally Advanced or Metastatic Cholangiocarcinoma (ProvIDHe) | Recruiting | SWE | ROU | NLD | ITA | IRL | GBR | FRA | ESP | DEU | CAN | BEL | AUT | AUS | 2 |
NCT04056910 | Phase II | Ivosidenib + Nivolumab | Ivosidenib (AG-120) With Nivolumab in IDH1 Mutant Tumors | Completed | USA | 0 |
NCT04088188 | Phase I | Cisplatin + Gemcitabine + Pemigatinib Cisplatin + Gemcitabine + Ivosidenib | Gemcitabine and Cisplatin With Ivosidenib or Pemigatinib for the Treatment of Unresectable or Metastatic Cholangiocarcinoma | Terminated | USA | 0 |
NCT06161974 | Phase II | Olutasidenib + Temozolomide | Study of Olutasidenib and Temozolomide in HGG | Not yet recruiting | USA | NLD | GBR | DEU | CAN | AUS | 0 |
NCT03953898 | Phase II | Olaparib | Using the Anticancer Drug Olaparib to Treat Relapsed/Refractory Acute Myeloid Leukemia or Myelodysplastic Syndrome With an Isocitrate Dehydrogenase (IDH) Mutation | Active, not recruiting | USA | 0 |
NCT05921760 | Phase Ib/II | Ipilimumab + Ivosidenib + Nivolumab | Ivosidenib, Nivolumab, and Ipilimumab Combination in Previously Treated Subjects With Nonresectable or Metastatic IDH1 Mutant Cholangiocarcinoma | Active, not recruiting | USA | GBR | 0 |
NCT04164901 | Phase III | Vorasidenib | Study of Vorasidenib (AG-881) in Participants With Residual or Recurrent Grade 2 Glioma With an IDH1 or IDH2 Mutation (INDIGO) | Active, not recruiting | USA | NLD | ITA | ISR | GBR | FRA | ESP | DEU | CHE | CAN | 1 |
NCT06127407 | Phase III | Ivosidenib | Ivosidenib in Participants With Locally Advanced or Metastatic Conventional Chondrosarcoma Untreated or Previously Treated With 1 Systemic Treatment Regimen (CHONQUER) | Recruiting | USA | CAN | BRA | AUS | 1 |