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Gene | BRAF |
Variant | G469V |
Impact List | missense |
Protein Effect | gain of function |
Gene Variant Descriptions | BRAF G469V is a hotspot mutation within the protein kinase domain of the Braf protein (UniProt.org). G469V results in increased Braf kinase activity and activation of downstream MEK and ERK in cell culture (PMID: 28947956, PMID: 26343582, PMID: 28783719), and in one of two cell lines, increased cell proliferation and cell viability compared to wild-type Braf (PMID: 29533785). |
Associated Drug Resistance | |
Category Variants Paths |
BRAF mutant BRAF act mut BRAF G469V BRAF mutant BRAF G469X BRAF G469V |
Transcript | NM_004333.6 |
gDNA | chr7:g.140781602C>A |
cDNA | c.1406G>T |
Protein | p.G469V |
Source Database | RefSeq |
Genome Build | GRCh38/hg38 |
Transcript | gDNA | cDNA | Protein | Source Database | Genome Build |
---|---|---|---|---|---|
XM_047420769.1 | chr7:g.140781602C>A | c.1406G>T | p.G469V | RefSeq | GRCh38/hg38 |
XM_005250045 | chr7:g.140781602C>A | c.1406G>T | p.G469V | RefSeq | GRCh38/hg38 |
NM_001354609.1 | chr7:g.140781602C>A | c.1406G>T | p.G469V | RefSeq | GRCh38/hg38 |
NM_004333.6 | chr7:g.140781602C>A | c.1406G>T | p.G469V | RefSeq | GRCh38/hg38 |
NM_001378474.1 | chr7:g.140781602C>A | c.1406G>T | p.G469V | RefSeq | GRCh38/hg38 |
NM_004333 | chr7:g.140781602C>A | c.1406G>T | p.G469V | RefSeq | GRCh38/hg38 |
NM_001354609.2 | chr7:g.140781602C>A | c.1406G>T | p.G469V | RefSeq | GRCh38/hg38 |
NM_001378468.1 | chr7:g.140781602C>A | c.1406G>T | p.G469V | RefSeq | GRCh38/hg38 |
NM_004333.5 | chr7:g.140781602C>A | c.1406G>T | p.G469V | RefSeq | GRCh38/hg38 |
NM_001378470.1 | chr7:g.140778000C>A | c.1406G>T | p.G469V | RefSeq | GRCh38/hg38 |
NM_001378467.1 | chr7:g.140781611C>A | c.1406G>T | p.G469V | RefSeq | GRCh38/hg38 |
Molecular Profile | Protein Effect | Treatment Approaches |
---|---|---|
BRAF G469V | gain of function | MEK inhibitor (Pan) MEK1 Inhibitor MEK2 Inhibitor |
BRAF G469V NRAS Q61K |