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Gene | BRAF |
Variant | V600E/K |
Impact List | missense |
Protein Effect | gain of function |
Gene Variant Descriptions | BRAF V600E/K indicates a mutation that results in the replacement of the valine (V) at amino acid 600 of the Braf protein by either a glutamate (E) or lysine (K). V600E/K mutations are hotspot mutations in Braf that result in increased Braf kinase activity (PMID: 15035987). |
Associated Drug Resistance | |
Category Variants Paths |
BRAF mutant BRAF act mut BRAF V600E/K BRAF mutant BRAF V600X BRAF V600E/K |
Molecular Profile | Protein Effect | Treatment Approaches |
---|---|---|
BRAF V600E/K | gain of function | BRAF Inhibitor MEK inhibitor (Pan) MEK1 Inhibitor MEK2 Inhibitor RAF Inhibitor (Pan) |
BRAF V600E/K PIK3CA wild-type | ||
BRAF V600E/K PTEN loss | ||
BRAF V600E/K CDKN2A loss RB1 pos |