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Gene | ALK |
Variant | C1237Y |
Impact List | missense |
Protein Effect | gain of function - predicted |
Gene Variant Descriptions | ALK C1237Y lies within the protein kinase domain of the Alk protein (UniProt.org). C1237Y results in both increased phosphorylation of Alk and proliferation, and has been demonstrated to confer resistance to Alk inhibitors in the context of EML4-ALK in culture (PMID: 38448512), and therefore, is predicted to lead to a gain of Alk protein function. |
Associated Drug Resistance | Y |
Category Variants Paths |
ALK mutant ALK act mut ALK C1237Y |
Transcript | NM_004304.5 |
gDNA | chr2:g.29214017C>T |
cDNA | c.3710G>A |
Protein | p.C1237Y |
Source Database | RefSeq |
Genome Build | GRCh38/hg38 |
Transcript | gDNA | cDNA | Protein | Source Database | Genome Build |
---|---|---|---|---|---|
NM_004304.5 | chr2:g.29214017C>T | c.3710G>A | p.C1237Y | RefSeq | GRCh38/hg38 |
Molecular Profile | Protein Effect | Treatment Approaches |
---|---|---|
ALK C1237Y | gain of function - predicted | |
EML4 - ALK ALK C1237Y | ||
EML4 - ALK ALK C1235R ALK C1237Y |