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Gene | BRAF |
Variant | D594E |
Impact List | missense |
Protein Effect | loss of function |
Gene Variant Descriptions | BRAF D594E lies within the protein kinase domain of the Braf protein (UniProt.org). D594E results in impaired Braf kinase activity, however, results in increased Mek and Erk phosphorylation in the presence of CRAF in cell culture (PMID: 28783719). |
Associated Drug Resistance | |
Category Variants Paths |
BRAF mutant BRAF D594X BRAF D594E BRAF mutant BRAF inact mut BRAF D594E |
Transcript | NM_004333.6 |
gDNA | chr7:g.140753353A>C |
cDNA | c.1782T>G |
Protein | p.D594E |
Source Database | RefSeq |
Genome Build | GRCh38/hg38 |
Transcript | gDNA | cDNA | Protein | Source Database | Genome Build |
---|---|---|---|---|---|
NM_001354609.1 | chr7:g.140753353A>C | c.1782T>G | p.D594E | RefSeq | GRCh38/hg38 |
NM_004333 | chr7:g.140753353A>C | c.1782T>G | p.D594E | RefSeq | GRCh38/hg38 |
NM_004333.6 | chr7:g.140753353A>C | c.1782T>G | p.D594E | RefSeq | GRCh38/hg38 |
NM_001378474.1 | chr7:g.140753353A>C | c.1782T>G | p.D594E | RefSeq | GRCh38/hg38 |
NM_001378468.1 | chr7:g.140753353A>C | c.1782T>G | p.D594E | RefSeq | GRCh38/hg38 |
NM_004333.5 | chr7:g.140753353A>C | c.1782T>G | p.D594E | RefSeq | GRCh38/hg38 |
NM_001354609.2 | chr7:g.140753353A>C | c.1782T>G | p.D594E | RefSeq | GRCh38/hg38 |
XM_005250045 | chr7:g.140753353A>C | c.1782T>G | p.D594E | RefSeq | GRCh38/hg38 |
Molecular Profile | Protein Effect | Treatment Approaches |
---|---|---|
BRAF D594E | loss of function | MEK inhibitor (Pan) MEK1 Inhibitor MEK2 Inhibitor |
BRAF D594E HRAS Q61L |