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| Drug Name | VT3989 |
| Trade Name | |
| Synonyms | VT-3989|VT 3989 |
| Drug Descriptions |
VT3989 inhibits the auto-palymitoylation of TEAD, which leads to impaired YAP function, potentially leading to inhibition of tumor growth (Cancer Res (2023) 83 (8_Supplement): CT006). |
| DrugClasses | |
| CAS Registry Number | NA |
| NCIT ID | C179669 |
| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| Ipilimumab + Nivolumab + VT3989 | Ipilimumab Nivolumab VT3989 | 0 | 1 |
| Osimertinib + VT3989 | Osimertinib VT3989 | 0 | 1 |
| VT3989 | VT3989 | 0 | 0 |