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Drug Name TAS-117
Trade Name
Synonyms TAS117|TAS 117
Drug Descriptions

TAS-117 is a selective allosteric inhibitor of Akt that inhibits Akt phosphorylation and downstream signaling, potentially leading to cytoxicity in tumor cells and decreased tumor growth (PMID: 24934808).

DrugClasses Akt Inhibitor (Pan) 21
CAS Registry Number 1402602-94-1
NCIT ID C178300

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Therapy Name Drugs Efficacy Evidence Clinical Trials
Futibatinib + TAS-117 Futibatinib TAS-117 0 0
TAS-117 TAS-117 4 1


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