Mubritinib
Drug Detail
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| Drug Name | Mubritinib |
| Trade Name | |
| Synonyms | TAK165|TAK 165|TAK-165 |
| Drug Descriptions |
Mubritinib (TAK-165) selectively inhibits ERBB2 (HER2), potentially resulting in oxidative stress, apoptosis (PMID: 31287994), decreased tumor cell viability (PMID: 34715459), and reduced tumor cell proliferation and tumor growth (PMID: 16771730). |
| DrugClasses | HER2 Inhibitor 44 |
| CAS Registry Number | 366017-09-6 |
| NCIT ID | C66212 |
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| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| Mubritinib | Mubritinib | 0 | 0 |
| Mubritinib + Sotorasib | Mubritinib Sotorasib | 0 | 0 |
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