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| Drug Name | LP-168 |
| Trade Name | |
| Synonyms | LP168|LP 168 |
| Drug Descriptions |
LP-168 is a selective BTK inhibitor with activity against wild-type BTK and BTK C481S, potentially inducing cytotoxicity in tumor cells and leading to antitumor activity (Blood (2023) 142 (Supplement 1): 416, Blood (2023) 142 (Supplement 1): 4400). |
| DrugClasses | BTK inhibitor 38 |
| CAS Registry Number | NA |
| NCIT ID | C202999 |
| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| LP-168 | LP-168 | 0 | 1 |
| LP-168 + Obinutuzumab | LP-168 Obinutuzumab | 0 | 1 |