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Drug Name DZD8586
Trade Name
Synonyms DZD-8586|DZD 8586
Drug Descriptions

DZD8586 is a non-covalent inhibitor of BTK and LYN that is blood-brain barrier-penetrant, which potentially induces tumor cell death and decreases tumor growth (Blood (2023) 142 (Supplement 1): 2822).

DrugClasses BTK inhibitor 37 LYN Inhibitor 4
CAS Registry Number NA
NCIT ID C200855

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Therapy Name Drugs Efficacy Evidence Clinical Trials
DZD8586 DZD8586 0 1


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