Missing content? – Request curation!
Request curation for specific Genes, Variants, or PubMed publications.
Have questions, comments, or suggestions? - Let us know!
Email us at : ckbsupport@genomenon.com
| Drug Name | TGRX-678 |
| Trade Name | |
| Synonyms | TGRX 678|TGRX678 |
| Drug Descriptions |
TGRX-678 inhibits BCR-ABL1 and ABL1 mutations including T315I, potentially resulting in decreased cell proliferation and inhibition of tumor growth (Blood (2023) 142 (Supplement 1): 2807). |
| DrugClasses | ABL1 Inhibitor 8 BCR-ABL Inhibitor 32 |
| CAS Registry Number | NA |
| NCIT ID | C202237 |
| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| Ponatinib + TGRX-678 | Ponatinib TGRX-678 | 0 | 0 |
| TGRX-678 | TGRX-678 | 0 | 1 |