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| Drug Name | Elenestinib |
| Trade Name | |
| Synonyms | BLU-263|BLU 263|BLU263 |
| Drug Descriptions |
Elenestinib (BLU-263) inhibits KIT D816V, which potentially leads to decreased cell proliferation (Blood (2022) 140 (Supplement 1): 6877–6878; NCI Drug Dictionary). |
| DrugClasses | KIT Inhibitor 57 |
| CAS Registry Number | 2505078-08-8 |
| NCIT ID | C180833 |
| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| Azacitidine + Elenestinib | Azacitidine Elenestinib | 0 | 1 |
| Elenestinib | Elenestinib | 0 | 2 |