Missing content? – Request curation!
Request curation for specific Genes, Variants, or PubMed publications.
Have questions, comments, or suggestions? - Let us know!
Email us at : ckbsupport@genomenon.com
| Drug Name | BAY3563254 |
| Trade Name | |
| Synonyms | BAY 3563254|225Ac-PSMA-Trillium |
| Drug Descriptions |
BAY3563254 comprises a PSMA inhibitor linked to the radionuclide Actinium-225, with an albumin domain for increased tumor uptake and a chelator for stable radiolabeling, which delivers radiation to PSMA-expressing tumor cells, potentially inhibiting tumor growth (Cancer Res (2024) 84 (7_Supplement): ND09). |
| DrugClasses | |
| CAS Registry Number | NA |
| NCIT ID | NA |
| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| BAY3563254 | BAY3563254 | 0 | 1 |