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| Drug Name | BBO-8520 |
| Trade Name | |
| Synonyms | BBO8520|BBO 8520 |
| Drug Descriptions |
BBO-8520 inhibits KRAS G12C in both the active and inactive states, which potentially decreases downstream signaling, cell viability, and tumor growth (PMID: 39642212). |
| DrugClasses | KRAS G12C inhibitor 36 |
| CAS Registry Number | 2893809-51-1 |
| NCIT ID | C205358 |
| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| BBO-10203 + BBO-8520 | BBO-10203 BBO-8520 | 0 | 0 |
| BBO-8520 | BBO-8520 | 0 | 1 |
| BBO-8520 + Pembrolizumab | BBO-8520 Pembrolizumab | 0 | 1 |