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| Drug Name | Lomonitinib |
| Trade Name | |
| Synonyms | ZE46 0134|ZE46-0134|ZE46 0134 |
| Drug Descriptions |
Lomonitinib (ZE46-0134) is an inhibitor of FLT3 and IRAK4, with activity against FLT3-ITD mutations and FLT3 F691L, which reduces downstream signaling and potentially inhibits tumor cell proliferation (Blood (2024) 144 (Supplement 1): 1396, NCI Drug Dictionary). |
| DrugClasses | FLT3 Inhibitor 69 IRAK4 Inhibitor 8 |
| CAS Registry Number | NA |
| NCIT ID | C215087 |
| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| Lomonitinib | Lomonitinib | 0 | 1 |