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Therapy Name | Lomonitinib |
Synonyms | |
Therapy Description |
Lomonitinib (ZE46-0134) is an inhibitor of FLT3 and IRAK4, with activity against FLT3-ITD mutations and FLT3 F691L, which reduces downstream signaling and potentially inhibits tumor cell proliferation (Blood (2024) 144 (Supplement 1): 1396, NCI Drug Dictionary). |