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| Drug Name | JI-101 |
| Trade Name | |
| Synonyms | CGI-1842 |
| Drug Descriptions |
JI-101 inhibits KDR (VEGFR2), PDGFR-beta (PDGFRB), and EphB4, resulting in anti-tumor activity (PMID: 26365907, PMID: 32336043). |
| DrugClasses | EPHB4 Inhibitor 6 PDGFR-beta Inhibitor 14 VEGFR2 Inhibitor 37 |
| CAS Registry Number | 900573-88-8 |
| NCIT ID | C82413 |
| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| Everolimus + JI-101 | Everolimus JI-101 | 0 | 0 |
| JI-101 | JI-101 | 0 | 0 |