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| Drug Name | Lonafarnib |
| Trade Name | Sarasar |
| Synonyms | SCH66336 |
| Drug Descriptions |
Lonafarnib (SCH66336) is a farnesyl transferase inhibitor, which alters post-translational modification and activation of Ras proteins (PMID: 25323927, PMID: 29285232). |
| DrugClasses | Farnesyltransferase Inhibitor 4 |
| CAS Registry Number | 193275-84-2 |
| NCIT ID | C1829 |
| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| Adagrasib + Lonafarnib | Adagrasib Lonafarnib | 0 | 0 |
| Docetaxel + Lonafarnib | Docetaxel Lonafarnib | 0 | 0 |
| Lonafarnib | Lonafarnib | 0 | 0 |
| Lonafarnib + Sotorasib | Lonafarnib Sotorasib | 0 | 0 |
| Lonafarnib + Tamoxifen | Lonafarnib Tamoxifen | 0 | 0 |