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| Drug Name | TGX-221 |
| Trade Name | |
| Synonyms | |
| Drug Descriptions |
TGX-221 is a selective inhibitor of PIK3CB which may inhibit transformation and proliferation of tumor cells (PMID: 15834429, PMID: 25473181, PMID: 31083328). |
| DrugClasses | PIK3CB inhibitor 8 |
| CAS Registry Number | 663619-89-4 |
| NCIT ID | NA |
| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| Ruxolitinib + TGX-221 | Ruxolitinib TGX-221 | 2 | 0 |
| TGX-221 | TGX-221 | 3 | 0 |