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Drug Detail
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| Drug Name | GSK3052230 |
| Trade Name | |
| Synonyms | FP-1039|HGS1036|GSK-3052230|GSK 3052230 |
| Drug Descriptions |
GSK3052230 (FP-1039) is an FGF ligand trap which prevents FGF1, FGF2, and FGF4 from binding corresponding receptors thereby preventing downstream signaling and activation (PMID: 26078430, PMID: 31065954, PMID: 31446228). |
| DrugClasses | |
| CAS Registry Number | 1631072-93-9 |
| NCIT ID | C77970 |
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| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| Carboplatin + GSK3052230 + Paclitaxel | Carboplatin GSK3052230 Paclitaxel | 1 | 0 |
| Cisplatin + Etoposide + GSK3052230 | Cisplatin Etoposide GSK3052230 | 1 | 0 |
| Cisplatin + GSK3052230 + Pemetrexed Disodium | Cisplatin GSK3052230 Pemetrexed Disodium | 0 | 0 |
| GSK3052230 | GSK3052230 | 4 | 1 |
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