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Drug Name | GSK126 |
Trade Name | |
Synonyms | GSK2816126|GSK-126 |
Drug Descriptions |
GSK126 selectively inhibits EZH2, resulting in decreased H3K27 tri-methylation, and potentially leading to decreased tumor cell proliferation and reduced tumor growth (PMID: 23051747, PMID: 25686104, PMID: 31471312). |
DrugClasses | EZH2 inhibitor 20 |
CAS Registry Number | 1346574-57-9 |
NCIT ID | C113334 |