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| Drug Name | Pipendoxifene |
| Trade Name | |
| Synonyms | ERA-923|ERA 923|ERA923 |
| Drug Descriptions |
Pipendoxifene (ERA-923) is a selective estrogen receptor modulator, which potently inhibits estrogen binding to Esr1 (ER alpha) in breast cancer cells (PMID: 11595711, PMID: 18279543). |
| DrugClasses | Hormone - Anti-estrogens 31 |
| CAS Registry Number | 198480-55-6 |
| NCIT ID | C1874 |
| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| Palbociclib + Pipendoxifene | Palbociclib Pipendoxifene | 0 | 0 |
| Pipendoxifene | Pipendoxifene | 0 | 0 |