Missing content? – Request curation!
Request curation for specific Genes, Variants, or PubMed publications.
Have questions, comments, or suggestions? - Let us know!
Email us at : ckbsupport@genomenon.com
| Drug Name | FRAX597 |
| Trade Name | |
| Synonyms | FRAX-597 |
| Drug Descriptions |
FRAX597 is a small-molecule inhibitor of the group I PAKs (PAK1, PAK2, and PAK3), which may result in decreased tumor growth (PMID: 23543898, PMID: 32186433, PMID: 32064922). |
| DrugClasses | PAK1 Inhibitor 11 |
| CAS Registry Number | 1286739-19-2 |
| NCIT ID | NA |
| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| FRAX597 | FRAX597 | 0 | 0 |
| FRAX597 + Sotorasib | FRAX597 Sotorasib | 0 | 0 |