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| Drug Name | MS417 |
| Trade Name | |
| Synonyms | |
| Drug Descriptions |
MS417 is a BET bromodomain inhibitor with specificity for BRD4, which may result in cell cycle arrest thereby inhibiting cell proliferation (PMID: 23950209, PMID: 22645123). |
| DrugClasses | BET Inhibitor (Pan) 33 |
| CAS Registry Number | 916489-36-6 |
| NCIT ID | NA |
| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| MS417 | MS417 | 0 | 0 |
| MS417 + Pictilisib | MS417 Pictilisib | 2 | 0 |