GSK-J4
Drug Detail
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| Drug Name | GSK-J4 |
| Trade Name | |
| Synonyms | |
| Drug Descriptions |
GSK-J4 is a specific inhibitor of KDM6, which results in increased H3K27 tri-methylation and induction of DNA damage response and cell death (PMID: 22842901, PMID: 26759175, PMID: 32525734, PMID: 32477122, PMID: 32514253). |
| DrugClasses | |
| CAS Registry Number | 1373423-53-0 |
| NCIT ID | NA |
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| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| GSK-J4 | GSK-J4 | 0 | 0 |
| GSK-J4 + PKF118-310 | GSK-J4 PKF118-310 | 0 | 0 |
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