PKF118-310
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| Drug Name | PKF118-310 |
| Trade Name | |
| Synonyms | |
| Drug Descriptions |
PKF118-310 inhibits KDM4A activity (PMID: 27767379) and the CTNNB1/TCF interaction, which results in apoptosis and anti-tumor activity (PMID: 19662654). |
| DrugClasses | CTNNB1 Inhibitor 27 KDM4 Inhibitor 4 |
| CAS Registry Number | NA |
| NCIT ID | NA |
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| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| GSK-J4 + PKF118-310 | GSK-J4 PKF118-310 | 0 | 0 |
| Imatinib + PKF118-310 | Imatinib PKF118-310 | 1 | 0 |
| PKF118-310 | PKF118-310 | 1 | 0 |
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