CX-6258
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| Drug Name | CX-6258 |
| Trade Name | |
| Synonyms | CX6258|CX 6258 |
| Drug Descriptions |
CX-6258 is an inhibitor of PIM1, PIM2, PIM3 and Histone H3-associated protein serine/threonine kinase (HASPIN), which may potentially result in antitumor activity (PMID: 24900437) and may overcome tumor resistance to RAF/MEK-inhibitors (PMID: 31882401). |
| DrugClasses | PIM Inhibitor (Pan) 10 |
| CAS Registry Number | 1202916-90-2 |
| NCIT ID | NA |
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| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| CX-5461 + CX-6258 | CX-5461 CX-6258 | 1 | 0 |
| CX-6258 | CX-6258 | 1 | 0 |
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