PKI-402
Drug Detail
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| Drug Name | PKI-402 |
| Trade Name | |
| Synonyms | |
| Drug Descriptions |
PKI-402 is a dual ATP-competitive mTOR/PI3K inhibitor, which leads to reduced downstream signaling, potentially resulting in decreased tumor growth (PMID: 20371716, PMID: 32585451). |
| DrugClasses | mTOR Inhibitor 51 PI3K Inhibitor (Pan) 42 |
| CAS Registry Number | NA |
| NCIT ID | NA |
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| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| H3B-5942 + PKI-402 | H3B-5942 PKI-402 | 0 | 0 |
| PKI-402 | PKI-402 | 2 | 0 |
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