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| Drug Name | H3B-5942 |
| Trade Name | |
| Synonyms | CS-0047696 |
| Drug Descriptions |
H3B-5942 is a selective estrogen receptor covalent antagonist, which antagonizes wild-type and mutant forms of estrogen receptor alpha, potentially resulting in decreased tumor cell proliferation and reduced tumor growth (PMID: 29991605). |
| DrugClasses | Hormone - Anti-estrogens 31 |
| CAS Registry Number | 2052128-15-9 |
| NCIT ID | NA |
| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| Abemaciclib + H3B-5942 | Abemaciclib H3B-5942 | 0 | 0 |
| AZD8055 + H3B-5942 | AZD8055 H3B-5942 | 0 | 0 |
| Everolimus + H3B-5942 | Everolimus H3B-5942 | 0 | 0 |
| H3B-5942 | H3B-5942 | 0 | 0 |
| H3B-5942 + Palbociclib | H3B-5942 Palbociclib | 0 | 0 |
| H3B-5942 + PF-04691502 | H3B-5942 PF-04691502 | 0 | 0 |
| H3B-5942 + PKI-402 | H3B-5942 PKI-402 | 0 | 0 |
| H3B-5942 + Ribociclib | H3B-5942 Ribociclib | 0 | 0 |
| H3B-5942 + Sirolimus | H3B-5942 Sirolimus | 0 | 0 |
| H3B-5942 + Temsirolimus | H3B-5942 Temsirolimus | 0 | 0 |