RVX2135
Drug Detail
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| Drug Name | RVX2135 |
| Trade Name | |
| Synonyms | |
| Drug Descriptions |
RVX2135 is a small molecule inhibitor of BET that binds to BRD2, BRD3, and BRD4, and may result in inhibition of cell proliferation, cell cycle arrest, and induced apoptosis (AACR; Cancer Res 2013;73(8 Suppl):Abstract nr LB-92, PMID: 24979794). |
| DrugClasses | BET Inhibitor (Pan) 33 |
| CAS Registry Number | NA |
| NCIT ID | NA |
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| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| AZ20 + RVX2135 | AZ20 RVX2135 | 0 | 0 |
| RVX2135 | RVX2135 | 0 | 0 |
| RVX2135 + VE-821 | RVX2135 VE-821 | 0 | 0 |
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