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Drug Name RVX2135
Trade Name
Synonyms
Drug Descriptions

RVX2135 is a small molecule inhibitor of BET that binds to BRD2, BRD3, and BRD4, and may result in inhibition of cell proliferation, cell cycle arrest, and induced apoptosis (AACR; Cancer Res 2013;73(8 Suppl):Abstract nr LB-92, PMID: 24979794).

DrugClasses BET Inhibitor (Pan) 32
CAS Registry Number NA
NCIT ID NA

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Therapy Name Drugs Efficacy Evidence Clinical Trials
AZ20 + RVX2135 AZ20 RVX2135 0 0
RVX2135 RVX2135 0 0
RVX2135 + VE-821 RVX2135 VE-821 0 0


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