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Drug Name | BETd-246 |
Trade Name | |
Synonyms | BET-d246 |
Drug Descriptions |
BETd-246 is a small molecule that induces degradation of Brd2, Brd3, and Brd4 proteins, leading to apoptosis of tumor cells (PMID: 28209615, PMID: 30797188). |
DrugClasses | BRD2 Inhibitor 1 BRD3 Inhibitor 2 BRD4 Inhibitor 10 |
CAS Registry Number | 2140289-17-2 |
NCIT ID | NA |
Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
---|---|---|---|
A-1155463 + BETd-246 | A-1155463 BETd-246 | 0 | 0 |
BETd-246 | BETd-246 | 0 | 0 |
BETd-246 + BM-1197 | BETd-246 BM-1197 | 0 | 0 |
BETd-246 + Navitoclax | BETd-246 Navitoclax | 0 | 0 |