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| Drug Name | BI 894999 |
| Trade Name | |
| Synonyms | BI894999|BI-894999 |
| Drug Descriptions |
BI 894999 is a bromodomain (BET) inhibitor with selective activity against BRD2/3/4 and BRDT, which may result in G1 arrest and apoptosis, and inhibition of tumor growth (Mol Cancer Ther 2015;14(12 Suppl 2):Abstract nr B79, PMID: 29491412). |
| DrugClasses | BET Inhibitor (Pan) 33 |
| CAS Registry Number | 1660117-38-3 |
| NCIT ID | C160257 |
| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| BI 894999 | BI 894999 | 0 | 1 |