Trigriluzole
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| Drug Name | Trigriluzole |
| Trade Name | |
| Synonyms | BHV-4157|BHV4157|Troriluzole |
| Drug Descriptions |
Trigriluzole (BHV-4157) is a small molecule inhibitor of the metabotropic glutamate receptor 1 (GRM1), which may prevent tumor growth (Journal of Clinical Oncology 36, no. 5_suppl, TPS80). |
| DrugClasses | |
| CAS Registry Number | 1926203-09-9 |
| NCIT ID | C142847 |
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| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| Ipilimumab + Nivolumab + Trigriluzole | Ipilimumab Nivolumab Trigriluzole | 0 | 1 |
| Nivolumab + Pembrolizumab + Trigriluzole | Nivolumab Pembrolizumab Trigriluzole | 0 | 1 |
| Trigriluzole | Trigriluzole | 0 | 1 |
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