GNE-049
Drug Detail
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| Drug Name | GNE-049 |
| Trade Name | |
| Synonyms | |
| Drug Descriptions |
GNE-049 inhibits the CBP and p300 bromodomains, resulting in decreased coactivator activity, and potentially leading to decreased tumor growth (PMID: 28819026). |
| DrugClasses | CBP/p300 inhibitor 13 |
| CAS Registry Number | 1936421-41-8 |
| NCIT ID | NA |
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| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| GNE-049 | GNE-049 | 0 | 0 |
| GNE-049 + Tegavivint | GNE-049 Tegavivint | 0 | 0 |
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