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| Drug Name | CORT125281 |
| Trade Name | |
| Synonyms | CORT-125281|CORT 125281|Exicorilant |
| Drug Descriptions |
Exicorilant (CORT125281) selectively antagonizes the glucocorticoid receptor (GR), resulting in decreased GR transcriptional activity (PMID: 28938459, PMID: 32369774). |
| DrugClasses | GR Antagonist 2 |
| CAS Registry Number | 1781244-77-6 |
| NCIT ID | C153309 |
| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| CORT125281 | CORT125281 | 0 | 0 |
| CORT125281 + Enzalutamide | CORT125281 Enzalutamide | 0 | 1 |