PLX51107
Drug Detail
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| Drug Name | PLX51107 |
| Trade Name | |
| Synonyms | PLX-51107|PLX 51107 |
| Drug Descriptions |
PLX51107 is a small molecule BET inhibitor, which binds to BET bromodomains in BRD2, BRD3, BRD4, and BRDT, potentially resulting in decreased tumor cell proliferation (PMID: 29386193, PMID: 31063649, PMID: 32717030). |
| DrugClasses | BET Inhibitor (Pan) 33 |
| CAS Registry Number | 1627929-55-8 |
| NCIT ID | C125739 |
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| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| Azacitidine + PLX51107 | Azacitidine PLX51107 | 0 | 1 |
| Dinaciclib + PLX51107 | Dinaciclib PLX51107 | 0 | 0 |
| PLX51107 | PLX51107 | 0 | 1 |
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