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Drug Name | PLX51107 |
Trade Name | |
Synonyms | PLX-51107|PLX 51107 |
Drug Descriptions |
PLX51107 is a small molecule BET inhibitor, which binds to BET bromodomains in BRD2, BRD3, BRD4, and BRDT, potentially resulting in decreased tumor cell proliferation (PMID: 29386193, PMID: 31063649, PMID: 32717030). |
DrugClasses | BET Inhibitor (Pan) 32 |
CAS Registry Number | 1627929-55-8 |
NCIT ID | C125739 |
Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
---|---|---|---|
Azacitidine + PLX51107 | Azacitidine PLX51107 | 0 | 1 |
Dinaciclib + PLX51107 | Dinaciclib PLX51107 | 0 | 0 |
PLX51107 | PLX51107 | 0 | 1 |