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| Drug Name | Grapiprant |
| Trade Name | |
| Synonyms | AT-001|CJ 023,423|RQ-07|AAT-007 |
| Drug Descriptions |
Grapiprant (AT-001) is a selective EP4 antagonist with analgesic and anti-inflammatory activity (PMID: 17495127, PMID: 28603634). |
| DrugClasses | |
| CAS Registry Number | 415903-37-6 |
| NCIT ID | C124131 |
| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| Grapiprant | Grapiprant | 0 | 0 |
| Grapiprant + Pembrolizumab | Grapiprant Pembrolizumab | 0 | 2 |