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| Drug Name | DFX117 |
| Trade Name | |
| Synonyms | DFX-117|DFX 117 |
| Drug Descriptions |
DFX117 is a dual inhibitor that blocks Met and selectively inhibits Pik3ca kinase activity, which potentially results in inhibition of cell proliferation, and induction of cell cycle arrest and apoptosis (PMID: 31060329, PMID: 28800461). |
| DrugClasses | MET Inhibitor 59 PIK3CA inhibitor 26 |
| CAS Registry Number | 2125500-60-7 |
| NCIT ID | NA |
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| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| DFX117 | DFX117 | 0 | 0 |
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