Missing content? – Request curation!
Request curation for specific Genes, Variants, or PubMed publications.
Have questions, comments, or suggestions? - Let us know!
Email us at : ckbsupport@genomenon.com
Gene | MAP2K1 |
Variant | Q56P |
Impact List | missense |
Protein Effect | gain of function |
Gene Variant Descriptions | MAP2K1 Q56P does not lie within any known functional domains of the Map2k1 protein (UniProt.org). Q56P confers a gain of function to the Map2k1 protein as indicated by increased kinase activity and the ability to transform cultured cells (PMID: 7651428, PMID: 22327936, PMID: 25351745) and increased proliferation in a competition assay (PMID: 36442478), and demonstrates resistance to some Mek and Braf inhibitors (PMID: 29753091). |
Associated Drug Resistance | Y |
Category Variants Paths |
MAP2K1 mutant MAP2K1 act mut MAP2K1 Q56P |
Transcript | NM_002755.4 |
gDNA | chr15:g.66435113A>C |
cDNA | c.167A>C |
Protein | p.Q56P |
Source Database | RefSeq |
Genome Build | GRCh38/hg38 |
Transcript | gDNA | cDNA | Protein | Source Database | Genome Build |
---|---|---|---|---|---|
NM_002755.3 | chr15:g.66435113A>C | c.167A>C | p.Q56P | RefSeq | GRCh38/hg38 |
NM_002755.4 | chr15:g.66435113A>C | c.167A>C | p.Q56P | RefSeq | GRCh38/hg38 |
XM_017022411.3 | chr15:g.66435113A>C | c.167A>C | p.Q56P | RefSeq | GRCh38/hg38 |
XM_017022411 | chr15:g.66435113A>C | c.167A>C | p.Q56P | RefSeq | GRCh38/hg38 |
NM_002755 | chr15:g.66435113A>C | c.167A>C | p.Q56P | RefSeq | GRCh38/hg38 |
XM_017022411.2 | chr15:g.66435113A>C | c.167A>C | p.Q56P | RefSeq | GRCh38/hg38 |
Molecular Profile | Protein Effect | Treatment Approaches |
---|---|---|
MAP2K1 Q56P | gain of function | MEK inhibitor (Pan) MEK1 Inhibitor |
BRAF V600E MAP2K1 Q56P | ||
BRAF V600E MAP2K1 Q56P NRAS Q61R | ||
MAP2K1 Q56P MAP2K1 H119Y MAP2K1 D351G |