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| Therapy Name | Pocenbrodib |
| Synonyms | |
| Therapy Description |
Pocenbrodib inhibits CREB binding protein (CBP) and p300, which potentially decreases proliferation of tumor cells expressing AR (Blood Cancer Discov (2024) 5 (2_Supplement): P33, NCI Drug Dictionary). |
| Drug Name | Trade Name | Synonyms | Drug Classes | Drug Description |
|---|---|---|---|---|
| Pocenbrodib | FT7051|FT 7051|FT7-051 | CBP/p300 inhibitor 13 | Pocenbrodib inhibits CREB binding protein (CBP) and p300, which potentially decreases proliferation of tumor cells expressing AR (Blood Cancer Discov (2024) 5 (2_Supplement): P33, NCI Drug Dictionary). |
| Molecular Profile | Indication/Tumor Type | Response Type | Therapy Name | Approval Status | Evidence Type | Efficacy Evidence | References |
|---|
| Clinical Trial | Phase | Therapies | Title | Recruitment Status | Covered Countries | Other Countries |
|---|---|---|---|---|---|---|
| NCT06785636 | Phase Ib/II | Pocenbrodib Abiraterone + Pocenbrodib Olaparib + Pocenbrodib lutetium Lu 177 vipivotide tetraxetan + Pocenbrodib | Open-Label Study of Pocenbrodib and in Combination With Abiraterone Acetate, Olaparib, or 177Lu-PSMA-617 (P300) | Recruiting | USA | 0 |
| NCT04575766 | Phase I | Pocenbrodib | A Study of FT-7051 in Men With MCRPC | Terminated | USA | 0 |