Missing content? – Request curation!
Request curation for specific Genes, Variants, or PubMed publications.
Have questions, comments, or suggestions? - Let us know!
Email us at : ckbsupport@genomenon.com
Drug Name | Pocenbrodib |
Trade Name | |
Synonyms | FT7051|FT 7051|FT7-051 |
Drug Descriptions |
Pocenbrodib inhibits CREB binding protein (CBP) and p300, which potentially decreases proliferation of tumor cells expressing AR (Blood Cancer Discov (2024) 5 (2_Supplement): P33, NCI Drug Dictionary). |
DrugClasses | CBP/p300 inhibitor 13 |
CAS Registry Number | NA |
NCIT ID | C178370 |
Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
---|---|---|---|
Abiraterone + Pocenbrodib | Abiraterone Pocenbrodib | 0 | 1 |
lutetium Lu 177 vipivotide tetraxetan + Pocenbrodib | Pocenbrodib lutetium Lu 177 vipivotide tetraxetan | 0 | 1 |
Olaparib + Pocenbrodib | Olaparib Pocenbrodib | 0 | 1 |
Pocenbrodib | Pocenbrodib | 0 | 2 |