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Therapy Name | IACS-6274 + Paclitaxel |
Synonyms | |
Therapy Description |
Limited information is currently available on IPN60090 (Apr, 2019). |
Drug Name | Trade Name | Synonyms | Drug Classes | Drug Description |
---|---|---|---|---|
IACS-6274 | IACS6274|IACS 6274|IPN60090|IPN-60090|IPN 60090 | Glutaminase Inhibitor 3 | IACS-6274 (IPN60090) inhibits glutaminase-1 (GLS1), which prevents the conversion of glutamine to glutamate, potentially resulting in decreased tumor cell proliferation (NCI Drug Dictionary). | |
Paclitaxel | Taxol | 7-Epipaclitaxel | Antimicrotubule Agent 14 BCL2 Family Inhibitor 6 | Taxol (paclitaxel) binds to tubulin to inhibit microtubule disassembly, which results in decreased cell division, and also binds to the anti-apoptotic factor Bcl-2, promoting apoptosis (NCI Drug Dictionary). |
Molecular Profile | Indication/Tumor Type | Response Type | Therapy Name | Approval Status | Evidence Type | Efficacy Evidence | References |
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Clinical Trial | Phase | Therapies | Title | Recruitment Status | Covered Countries | Other Countries |
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NCT03894540 | Phase I | IACS-6274 IACS-6274 + Pembrolizumab IACS-6274 + Paclitaxel | A Phase I, Dose Escalation and Dose Expansion Study of IPN60090 in Patients With Advanced Solid Tumours | Terminated | USA | 0 |