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| Drug Name | ZB716 |
| Trade Name | |
| Synonyms | ZB 716|ZB-716|Borestrant |
| Drug Descriptions |
ZB716 is a selective estrogen receptor degrader (SERD) that may inhibit growth of ESR1 (ER alpha)-positive tumor cells and decrease tumor growth (PMID: 29467940). |
| DrugClasses | Hormone - Anti-estrogens 31 |
| CAS Registry Number | 1853279-29-4 |
| NCIT ID | C179265 |
| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| Palbociclib + ZB716 | Palbociclib ZB716 | 0 | 1 |
| ZB716 | ZB716 | 0 | 1 |